

HC067047 Hydrochloride(883031-03-6 free base)
CAS No. 1481646-76-7
HC067047 Hydrochloride(883031-03-6 free base) ( —— )
产品货号. M23636 CAS No. 1481646-76-7
HC-067047 盐酸盐是一种有效的选择性 TRPV4 拮抗剂。
纯度: >98% (HPLC)






规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥2446 | 有现货 |
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10MG | ¥3669 | 有现货 |
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25MG | ¥6051 | 有现货 |
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50MG | ¥8505 | 有现货 |
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100MG | ¥11502 | 有现货 |
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500MG | ¥22923 | 有现货 |
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1G | 获取报价 | 有现货 |
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生物学信息
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产品名称HC067047 Hydrochloride(883031-03-6 free base)
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述HC-067047 盐酸盐是一种有效的选择性 TRPV4 拮抗剂。
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产品描述HC-067047 hydrochloride is a potent and selective TRPV4 antagonist. HC-067047 hydrochloride reversibly inhibited currents through the human, rat, and mouse TRPV4 orthologs with IC50 values of 486 nM, 133nM, and 17 nM, respectively.
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体外实验——
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体内实验——
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同义词——
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通路Membrane Transporter/Ion Channel
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靶点TRP/TRPV Channel
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受体TRPV4
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研究领域——
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适应症——
化学信息
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CAS Number1481646-76-7
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分子量507.98
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分子式C26H29ClF3N3O2
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纯度>98% (HPLC)
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溶解度——
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SMILESO=C(C1=C(C)N(CCCN2CCOCC2)C(C3=CC=CC=C3)=C1)NC4=CC=CC(C(F)(F)F)=C4.[H]Cl
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Xing Y , Ming J , Liu T , et al. Decreased Expression of TRPV4 Channels in HEI-OC1 Cells Induced by High Glucose Is Associated with Hearing Impairment[J]. Yonsei medical journal, 2018, 59(9).
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